Gianluca SBARDELLA

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Antonello MaiProfessore di Chimica Farmaceutica, Sapienza Università di RomaDirección de correo verificada de uniroma1.it
Sabrina CASTELLANOUniversità di SalernoDirección de correo verificada de unisa.it
Rino RagnoSapienza Università di Roma Diaprtimento di Chimica e Tecnologie del FarmacoDirección de correo verificada de uniroma1.it
Ettore NovellinoDipartimento di Farmacia, Università degli Studi di Napoli Federico IIDirección de correo verificada de unina.it
Dante Rotili, PhDProfessor of Medicinal Chemistry, "Sapienza" University of RomeDirección de correo verificada de uniroma1.it
Lucia Altucci, MD, PhDSeconda Università di NapoliDirección de correo verificada de unina2.it
Alessandra TOSCODepartment of Pharmacy, University of SalernoDirección de correo verificada de unisa.it
Donatella RescignoPhD Student, University of SalernoDirección de correo verificada de unisa.it
Sergio ValenteAssociate Professor, Sapienza University RomeDirección de correo verificada de uniroma1.it
Sandro CosconatiFull Professor of Medicinal Chemistry, University of Campania "Luigi Vanvitelli"Dirección de correo verificada de unicampania.it
Enzo TramontanoProfessore Ordinario di Microbiologia, Dipartimento di Scienze della Vita e dell'Ambiente, Università di CagliariDirección de correo verificada de unica.it
Maurizio C. CapogrossiJohns Hopkins University and National Institute on Aging, National Institutes of HealthDirección de correo verificada de jhu.edu
Carlo GaetanoLaboratorio di Epigenetica-Istituti Clinici Scientifici Maugeri, Pavia, Italy.Dirección de correo verificada de icsmaugeri.it
Giovanni GrecoProfessor of Medicinal Chemistry, Università di Napoli Federico IIDirección de correo verificada de unina.it
roberta loddoUniversità di Cagliari, Dipartimento di Scienze BiomedicheDirección de correo verificada de unica.it
Marco MiceliPost-Doc CEINGE-Biotecnologie Avanzate s.c.ar.l. Federico II NapoliDirección de correo verificada de ceinge.unina.it
Jose L. Medina-FrancoUniversidad Nacional Autonoma de Mexico (UNAM)Dirección de correo verificada de unam.mx
Andrea PintoDepartment of Food, Environmental and Nutritional Sciences - DeFENS, University of MilanDirección de correo verificada de unimi.it
Amodio Luca BalzanoAptuit, an Evotec CompanyDirección de correo verificada de evotec.com
Corrado SpadaforaInstitute of Translational Pharmacology, CNR National Research Council of ItalyDirección de correo verificada de ift.cnr.it

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Gianluca SBARDELLA

Dipartimento di Farmacia, Università di Salerno

Dirección de correo verificada de unisa.it

Medicinal Chemistry epigenetics Chemical Biology drug discovery


Título Ordenar por citas Ordenar por año Ordenar por título	Citado por Citado por	Año
Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees A Spannhoff, YK Kim, NJM Raynal, V Gharibyan, MB Su, YY Zhou, J Li, ... EMBO reports 12 (3), 238-243, 2011	230	2011
Synthesis and Biochemical Evaluation of Δ²-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors S Castellano, D Kuck, M Viviano, J Yoo, F López-Vallejo, P Conti, ... Journal of medicinal chemistry 54 (21), 7663-7677, 2011	199	2011
Arginine demethylation of G3BP1 promotes stress granule assembly WC Tsai, S Gayatri, LC Reineke, G Sbardella, MT Bedford, RE Lloyd Journal of Biological Chemistry 291 (43), 22671-22685, 2016	179	2016
Epigenetic multiple ligands: mixed histone/protein methyltransferase, acetyltransferase, and class III deacetylase (sirtuin) inhibitors A Mai, D Cheng, MT Bedford, S Valente, A Nebbioso, A Perrone, ... Journal of medicinal chemistry 51 (7), 2279-2290, 2008	164	2008
5-Alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4(3H)-ones: Novel Potent and Selective Dihydro-alkoxy-benzyl-oxopyrimidine Derivatives A Mai, M Artico, G Sbardella, S Massa, E Novellino, G Greco, AG Loi, ... Journal of Medicinal Chemistry 42 (4), 619-627, 1999	162	1999
Dihydro(alkylthio)(naphthylmethyl)oxopyrimidines: Novel Non-Nucleoside Reverse Transcriptase Inhibitors of the S-DABO Series A Mai, M Artico, G Sbardella, S Quartarone, S Massa, AG Loi, A De Montis, ... Journal of Medicinal Chemistry 40 (10), 1447-1454, 1997	162	1997
Small-molecule inhibitors of histone acetyltransferase activity: identification and biological properties A Mai, D Rotili, D Tarantino, P Ornaghi, F Tosi, C Vicidomini, G Sbardella, ... Journal of medicinal chemistry 49 (23), 6897-6907, 2006	161	2006
Preparation and anti-HIV-1 activity of Thio Analogues of Dichydroalkoxybenzyloxopyrimidines A Mai, M Artico, G Sbardella, S Massa, AG Loi, E Tramontano, P Scano, ... Journal of medicinal chemistry 38 (17), 3258-3263, 1995	141	1995
Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2, 6-difluorophenyl) alkyl]-3, 4-dihydro-5-alkylpyrimidin-4 … A Mai, G Sbardella, M Artico, R Ragno, S Massa, E Novellino, G Greco, ... Journal of medicinal chemistry 44 (16), 2544-2554, 2001	137	2001
Identification of long chain alkylidenemalonates as novel small molecule modulators of histone acetyltransferases G Sbardella, S Castellano, C Vicidomini, D Rotili, A Nebbioso, M Miceli, ... Bioorganic & medicinal chemistry letters 18 (9), 2788-2792, 2008	133	2008
Small molecule inhibitors of histone arginine methyltransferases: homology modeling, molecular docking, binding mode analysis, and biological evaluations R Ragno, S Simeoni, S Castellano, C Vicidomini, A Mai, A Caroli, ... Journal of medicinal chemistry 50 (6), 1241-1253, 2007	131	2007
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1 S Castellano, D Kuck, M Sala, E Novellino, F Lyko, G Sbardella Journal of medicinal chemistry 51 (7), 2321-2325, 2008	122	2008
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart C Colussi, J Rosati, S Straino, F Spallotta, R Berni, D Stilli, S Rossi, ... Proceedings of the National Academy of Sciences 108 (7), 2795-2800, 2011	121	2011
Computer-aided design, synthesis, and anti-HIV-1 activity in vitro of 2-alkylamino-6-[1-(2, 6-difluorophenyl) alkyl]-3, 4-dihydro-5-alkylpyrimidin-4 (3 H)-ones as novel potent … R Ragno, A Mai, G Sbardella, M Artico, S Massa, C Musiu, M Mura, ... Journal of medicinal chemistry 47 (4), 928-934, 2004	117	2004
p300/CBP-associated factor selectively regulates the extinction of conditioned fear W Wei, CM Coelho, X Li, R Marek, S Yan, S Anderson, D Meyers, ... Journal of Neuroscience 32 (35), 11930-11941, 2012	103	2012
3-(4-Aroyl-1 H-pyrrol-2-yl)-N-hydroxy-2-propenamides, a new class of synthetic histone deacetylase inhibitors S Massa, A Mai, G Sbardella, M Esposito, R Ragno, P Loidl, G Brosch Journal of medicinal chemistry 44 (13), 2069-2072, 2001	102	2001
The emerging role of lysine methyltransferase SETD8 in human diseases C Milite, A Feoli, M Viviano, D Rescigno, A Cianciulli, AL Balzano, A Mai, ... Clinical epigenetics 8, 1-15, 2016	99	2016
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases A Mai, D Rotili, D Tarantino, A Nebbioso, S Castellano, G Sbardella, ... Bioorganic & medicinal chemistry letters 19 (4), 1132-1135, 2009	99	2009
Novel 3, 5-bis (bromohydroxybenzylidene) piperidin-4-ones as coactivator-associated arginine methyltransferase 1 inhibitors: enzyme selectivity and cellular activity D Cheng, S Valente, S Castellano, G Sbardella, R Di Santo, R Costi, ... Journal of medicinal chemistry 54 (13), 4928-4932, 2011	91	2011
A New Facile and Expeditious Synthesis of N-Hydroxy-N′-Phenyloctanediamjde, a Potent Inducer of Terminal Cytodifferecntiation A Mai, M Esposito, G Sbardella, S Massa Organic Preparations and Procedures International 33 (4), 391-394, 2001	90	2001

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